I. Basic InformationProject | DetailsEnglish Name | RelugolixChinese Name | RuilugolixCAS Number | 737789-87-6 NCBIChemical Name | N-(4-{1-[(2,6-Difluorophenyl)methyl]-5-[(dimethylamino)methyl]-3-(6-m…
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I. Basic InformationItem | DetailsEnglish Name | Topiroxostat; FYX-051; TOPILORIC (Trade Name)Chinese Name | TopiroxostatCAS Number | 577778-58-6Chemical Name | 5-(2-cyano-4-pyridinyl)-3-(4-pyridinyl)…
I. Basic InformationItem | DetailsEnglish Name | Abemaciclib; Verzenio (trade name)Chinese Name | AbemaciclibCAS Number | 1231929-97-7Chemical Name | N-[5-[(4-ethyl-1-piperazinyl)methyl]-2-pyridinyl]-…
I. Basic InformationItem | DetailsEnglish Name | Vonoprazan fumarate; Takecab (trade name)Chinese Name | Vonoprazan fumarateCAS Number | 1260141-27-2 (fumarate); 1026256-79-0 (free base)Chemical Name …
I. Basic InformationItem DetailsEnglish Name VericiguatChinese Name 维立西呱 (Weiliciguat)Chemical Name Methyl {4,6-diamino-2-[5-fluoro-1-[(2-fluorobenzyl)-1H-pyrazolo[3,4-b]pyridin-3-yl]pyrimidin-5-yl}ca…
I. Basic InformationItem | DetailsEnglish Full Name | Benzenesulfonamide, 5-[(2,4-diamino-5-pyrimidinyl)oxy]-2-methoxy-4-(1-methylethyl)-, 2-hydroxy-1,2,3-propanetricarboxylate (1:1)Chinese Name | 5-[…
Basic InformationItem | DetailsEnglish Name | Fezolinetant; Veozah (Trade Name)Chinese Name | FezolinetantCAS Number | 1229705-11-1Chemical Name | (4-Fluorophenyl)[(8R)-8-methyl-3-(3-methyl-1,2,4-thia…
Physicochemical Properties (Sodium Salt)Appearance: White to off-white/pale yellow powder;Solubility: Easily soluble in water (approximately 100 mg/mL, pH 7.0), soluble in methanol and ethanol, slight…
Core Mechanism of Action and ResistanceMechanism of ActionIt specifically binds to the catalytic core of HIV integrase, inhibiting the strand transfer reaction (a key step in HIV replication), prevent…
Mechanism of Action and ResistanceMechanism: Inhibits the strand transfer reaction of HIV integrase, preventing viral DNA integration into the host genome and blocking viral replication.Resistance:…
PharmacokineticsAbsorption: Oral bioavailability is approximately 30%, and absorption is not affected by food. The time to reach peak concentration (Tmax) is approximately 2 hours.Distribution: Plasma…
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